Basic Information
ID: ALA4260475
Type: ADME
Description: Inhibition of human CYP2E1 expressed in baculosomes at 1 uM using EOMCC as substrate preincubated for 20 mins followed by substrate and NADP+ addition and measured after 30 mins by fluorescence assay
Format: BAO_0000019
Organism: Homo sapiens
Target: Cytochrome P450 2E1(ALA5281)
Document: ALA4257568
Inhibition of human CYP2E1 expressed in baculosomes at 1 uM using EOMCC as substrate preincubated for 20 mins followed by substrate and NADP+ addition and measured after 30 mins by fluorescence assay: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA4260475
Inhibition
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 151.16 | 1.35 | 1.35 |
| 332.34 | 1.18 | 1.18 |
| 449.40 | 0.97 | 0.97 |
| 463.42 | 1.36 | 1.36 |