Basic Information
ID: ALA4264842
Type: Binding
Description: Binding affinity to partial length wild type human EGFR (R669 to V1011 residues) expressed in bacterial expression system assessed as fraction of unbound kinase to substrate at 0.1 uM after 1 hr by KinomeScan assay
Format: BAO_0000019
Organism: Homo sapiens
Target: Epidermal growth factor receptor erbB1(ALA203)
Document: ALA4261615
Binding affinity to partial length wild type human EGFR (R669 to V1011 residues) expressed in bacterial expression system assessed as fraction of unbound kinase to substrate at 0.1 uM after 1 hr by KinomeScan assay: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA4264842
Activity
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 459.41 | 4.43 | 4.43 |
| 501.49 | 5.56 | 5.56 |
| 538.31 | 5.19 | 5.19 |
| 473.44 | 4.74 | 4.74 |