Basic Information
ID: ALA4264848
Type: Binding
Description: Binding affinity to full length wild type human GSK3beta (M1 to T433 residues) expressed in mammalian expression system assessed as fraction of unbound kinase to substrate at 0.1 uM after 1 hr by KinomeScan assay
Format: BAO_0000019
Organism: Homo sapiens
Target: Glycogen synthase kinase-3 beta(ALA262)
Document: ALA4261615
Binding affinity to full length wild type human GSK3beta (M1 to T433 residues) expressed in mammalian expression system assessed as fraction of unbound kinase to substrate at 0.1 uM after 1 hr by KinomeScan assay: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA4264848
Activity
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 459.41 | 4.43 | 4.43 |
| 501.49 | 5.56 | 5.56 |
| 538.31 | 5.19 | 5.19 |
| 473.44 | 4.74 | 4.74 |