Basic Information
ID: ALA4266824
Type: Binding
Description: Displacement of [3H]-T0901317 from recombinant human His-SUMO-tagged RORgamma LBD (265 to 518 residues) expressed in Escherichia coli BL21(DE3) at 1 uM after 1 hr by scintillation proximity assay
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA4266824
Inhibition
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 374.89 | 6.97 | 6.97 |
| 349.24 | 4.93 | 4.93 |
| 333.24 | 5.95 | 5.95 |
| 368.67 | 6.00 | 6.00 |
| 342.80 | 5.03 | 5.03 |
| 328.20 | 5.29 | 5.29 |
| 363.36 | 5.07 | 5.07 |
| 367.24 | 5.54 | 5.54 |
| 354.90 | 6.60 | 6.60 |
| 449.80 | 6.92 | 6.92 |
| 367.68 | 6.61 | 6.61 |
| 334.23 | 5.35 | 5.35 |
| 356.21 | 4.67 | 4.67 |