Assay Report Card

Basic Information

ID: ALA4267185

Type: Binding

Description: Inhibition of human GAT2 expressed in CHO cells assessed as reduction in [3H]GABA uptake at 100 uM after 20 mins by liquid scintillation counting analysis relative to control

Organism: Homo sapiens

Cell type: CHO

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
133.12-0.24-0.24
141.170.220.22
129.160.050.05
143.190.440.44
131.13-1.22-1.22
156.140.100.10
129.160.050.05
143.190.440.44