Basic Information
ID: ALA4270047
Type: Binding
Description: Inhibition of KDM6A (880 to 1401 residues) (unknown origin) using H3 ( 21 to 44 residues) K27me3 as substrate preincubated for 15 min followed by substrate addition measured after 15 mins by FDH-coupled demethylase assay
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA4270047
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 389.46 | 3.03 | 3.03 |
| 396.45 | 1.65 | 1.65 |
| 432.51 | 1.41 | 1.41 |