Basic Information
ID: ALA4272097
Type: Binding
Description: Inhibition of recombinant human His-tagged BRPF1 using biotinylated H4(1 to 21)K5/8/12/16Ac peptide as substrate after 30 mins by AlphaScreen assay
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA4272097
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 456.57 | 2.59 | 2.59 |
| 486.59 | 2.07 | 2.07 |
| 408.46 | 2.10 | 2.10 |
| 474.54 | 1.66 | 1.66 |
| 529.62 | 1.86 | 1.86 |
| 391.43 | 1.88 | 1.88 |
| 431.50 | 2.78 | 2.78 |
| 450.54 | 3.12 | 3.12 |
| 469.49 | 3.28 | 3.28 |
| 416.46 | 0.11 | 0.11 |
| 512.63 | 2.92 | 2.92 |
| 465.51 | 3.49 | 3.49 |
| 449.44 | 3.43 | 3.43 |
| 417.46 | 1.90 | 1.90 |
| 190.20 | 0.24 | 0.24 |
| 375.39 | 2.15 | 2.15 |
| 334.45 | 3.23 | 3.23 |
| 511.60 | 2.16 | 2.16 |
| 446.43 | 3.11 | 3.11 |
| 336.46 | 2.13 | 2.13 |
| 343.77 | 4.38 | 4.38 |
| 482.61 | 2.91 | 2.91 |
| 374.40 | 2.56 | 2.56 |
| 337.47 | 2.91 | 2.91 |
| 431.50 | 2.99 | 2.99 |
| 485.56 | 1.91 | 1.91 |
| 393.38 | 1.61 | 1.61 |
| 470.60 | 2.94 | 2.94 |
| 391.43 | 2.01 | 2.01 |
| 462.43 | 2.34 | 2.34 |
| 336.42 | 2.77 | 2.77 |
| 488.57 | 2.05 | 2.05 |
| 484.58 | 1.75 | 1.75 |
| 461.47 | 3.30 | 3.30 |
| 481.53 | 4.65 | 4.65 |
| 496.63 | 3.69 | 3.69 |
| 433.92 | 2.42 | 2.42 |
| 389.42 | 1.63 | 1.63 |
| 337.47 | 2.79 | 2.79 |
| 494.96 | 1.54 | 1.54 |
| 410.47 | 2.34 | 2.34 |
| 431.50 | 3.00 | 3.00 |
| 377.47 | 1.70 | 1.70 |
| 391.43 | 1.80 | 1.80 |
| 527.65 | 3.01 | 3.01 |
| 484.58 | 1.98 | 1.98 |
| 435.46 | 2.83 | 2.83 |
| 467.43 | 3.57 | 3.57 |
| 348.47 | 3.48 | 3.48 |
| 431.50 | 2.50 | 2.50 |
| 401.47 | 2.90 | 2.90 |
| 334.44 | 3.49 | 3.49 |
| 347.37 | 3.81 | 3.81 |
| 470.60 | 2.84 | 2.84 |
| 345.47 | 3.23 | 3.23 |
| 492.99 | 2.69 | 2.69 |
| 556.60 | 2.11 | 2.11 |
| 428.54 | 0.41 | 0.41 |