Assay Report Card

Basic Information

ID: ALA4272105

Type: Binding

Description: Inhibition of human GST-tagged BRD4 BD1 (44 to 170 residues) expressed in Escherichia coli BL21 using biotinylated H4(1 to 21)K5/8/12/16Ac peptide as substrate after 30 mins by AlphaScreen assay

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
486.592.072.07
343.774.384.38
348.473.483.48