Basic Information
ID: ALA4275379
Type: Binding
Description: Inhibition of 20S proteasome beta5 subunit in human Jurkat cell lysate using Suc-LLVY-AMC as substrate pretreated for 30 mins followed by substrate addition and measured after 60 mins by fluorescence assay
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA4275379
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 719.92 | 2.58 | 2.58 |
| 490.60 | 2.61 | 2.61 |
| 474.60 | 2.99 | 2.99 |
| 495.02 | 3.25 | 3.25 |
| 556.66 | 3.77 | 3.77 |
| 472.58 | 2.74 | 2.74 |
| 508.62 | 3.19 | 3.19 |
| 426.55 | 2.05 | 2.05 |
| 508.62 | 3.19 | 3.19 |
| 538.64 | 3.16 | 3.16 |
| 418.49 | 1.57 | 1.57 |
| 356.42 | 0.55 | 0.55 |
| 474.60 | 2.99 | 2.99 |
| 410.51 | 1.58 | 1.58 |
| 444.53 | 1.96 | 1.96 |
| 424.54 | 1.98 | 1.98 |
| 458.56 | 2.35 | 2.35 |
| 466.62 | 2.98 | 2.98 |
| 538.64 | 3.16 | 3.16 |
| 474.60 | 2.99 | 2.99 |
| 384.47 | 1.03 | 1.03 |
| 459.59 | 2.17 | 2.17 |
| 474.60 | 2.99 | 2.99 |
| 488.63 | 3.38 | 3.38 |
| 460.57 | 2.60 | 2.60 |
| 460.57 | 2.60 | 2.60 |