Assay Report Card

Basic Information

ID: ALA4275389

Type: Binding

Description: Inhibition of 20S proteasome beta5 subunit in human MCF7 cells using Suc-LLVY-AMC as substrate pretreated for 1 hr followed by compound washout and cell lysis prior to substrate addition measured after 1 hr by fluorescence assay

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
474.602.992.99
472.582.742.74
508.623.193.19
538.643.163.16
418.491.571.57
474.602.992.99
446.542.212.21
444.531.961.96
458.562.352.35
538.643.163.16
474.602.992.99
474.602.992.99
460.572.602.60
460.572.602.60