Assay Report Card

Basic Information

ID: ALA4305047

Type: Binding

Description: Inhibition of human N-terminal GST-tagged TNKS1 (1001 to 1327 residues) expressed in baculovirus infected Sf9 insect cells at 500 nM using histone as substrate measured after 1 hr by horseradish peroxidase-coupled chemiluminescence assay relative to control

Organism: Homo sapiens

Cell type: Sf9

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
434.472.352.35
493.523.243.24
483.412.672.67
495.502.352.35
455.472.532.53