Assay Report Card

Basic Information

ID: ALA4306967

Type: Binding

Description: Inhibition of N-terminal GST-tagged human NSD2 catalytic domain (941 to 1240 amino acids) expressed in Escherichia coli assessed as enzyme remaining activity at 50 uM pre-incubated for 15 mins followed by AdoMet addition and measured after 1 hr by luminescence method relative to control

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
507.550.490.49