Inhibition of human KGA (63 to 669 residues) preincubated for 15 mins using 50 mM glutamine as substrate by resorufin dye based assay

Basic Information

ID: ALA4309435

Type: Binding

Description: Inhibition of human KGA (63 to 669 residues) preincubated for 15 mins using 50 mM glutamine as substrate by resorufin dye based assay

Format: BAO_0000357

Organism: Homo sapiens

Target: Glutaminase kidney isoform, mitochondrial(ALA2146302)

Document: ALA4308839

Inhibition of human KGA (63 to 669 residues) preincubated for 15 mins using 50 mM glutamine as substrate by resorufin dye based assay: 1

Associated Items: Associated Bioactivities Associated Compounds

Activity Charts

Bioactivity

Activity Types for Assay ALA4309435

IC50

Total(15)

Parent Molecular Weight	ALogP	Polar Surface Area
412.48	1.74	1.74
411.49	2.35	2.35
454.56	2.27	2.27
508.53	3.16	3.16
459.51	2.49	2.49
445.94	3.00	3.00
412.48	1.74	1.74
454.56	2.27	2.27
525.51	3.25	3.25
436.55	2.19	2.19
525.51	3.25	3.25
520.54	3.30	3.30
471.47	2.89	2.89
411.49	2.35	2.35
508.53	3.16	3.16

Parent Molecular Weight

ALogP

Polar Surface Area

412.48

1.74

411.49

2.35

454.56

2.27

508.53

3.16

459.51

2.49

445.94

3.00

412.48

1.74

454.56

2.27

525.51

3.25

436.55

2.19

525.51

3.25

520.54

3.30

471.47

2.89