Assay Report Card

Basic Information

ID: ALA4310116

Type: Binding

Description: Inhibition of BRD4 bromodomain 1 in human A549 cells assessed as reduction in TNFalpha-induced NFkappaB transcription at 10 uM after 8 hrs by bright-glo luciferase reporter gene assay relative to control

Organism: Homo sapiens

Cell type: A549

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
442.545.435.43