Assay Report Card

Basic Information

ID: ALA4310249

Type: Binding

Description: Positive allosteric modulation of GABA-A alpha1beta3gamma2S receptor (unknown origin) expressed in Xenopus laevis oocytes assessed as increase in GABA-induced chloride current up to 100 uM after 15 mins at -70 mV holding potential by two-microelectrode voltage clamp method relative to control

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
274.543.783.78
234.343.793.79
191.663.583.58
214.094.014.01
212.083.923.92
255.102.782.78
191.663.583.58
212.083.923.92
255.102.782.78
255.102.782.78
237.093.813.81
212.083.923.92