Basic Information
ID: ALA4310278
Type: Binding
Description: Negative allosteric modulation of alpha4beta2 nAChR (unknown origin) expressed in Xenopus laevis oocytes assessed as decrease in acetylcholine-induced channel current at 100 uM at -70 mV holding potential by two-microelectrode voltage clamp method relative to control
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA4310278
Inhibition
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 237.09 | 3.81 | 3.81 |
| 212.08 | 3.92 | 3.92 |