Inhibition of recombinant human N-terminal His-tagged POP (2 to 710 residues) expressed in SF21 cells using Z-Gly-Pro-AMC as substrate incubated for 5...

Basic Information

ID: ALA4316407

Type: Binding

Description: Inhibition of recombinant human N-terminal His-tagged POP (2 to 710 residues) expressed in SF21 cells using Z-Gly-Pro-AMC as substrate incubated for 5 to 10 mins followed by substrate addition and measured for 30 mins by fluorescence based assay

Format: BAO_0000219

Organism: Homo sapiens

Cell type: Sf21

Target:  Prolyl endopeptidase(ALA3202)

Document:  ALA4312033

Inhibition of recombinant human N-terminal His-tagged POP (2 to 710 residues) expressed in SF21 cells using Z-Gly-Pro-AMC as substrate incubated for 5 to 10 mins followed by substrate addition and measured for 30 mins by fluorescence based assay: 1

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
232.281.881.88
294.09
389.25
275.281.721.72
368.29
410.32
386.28
353.27
371.26
293.271.861.86
275.281.911.91
250.272.022.02
401.29
428.31
252.05
276.10
440.35
399.37
383.30
257.291.771.77