Inhibition of human BTK assessed as remaining kinase activity at 1 uM using Cdc2 peptide KVEKIGEGTYGVVYK substrate and [gamma-33P]-ATP incubated for 4...

Basic Information

ID: ALA4321379

Type: Binding

Description: Inhibition of human BTK assessed as remaining kinase activity at 1 uM using Cdc2 peptide KVEKIGEGTYGVVYK substrate and [gamma-33P]-ATP incubated for 40 mins by radiometric protein kinase assay

Format: BAO_0000357

Organism: Homo sapiens

Target:  Tyrosine-protein kinase BTK(ALA5251)

Document:  ALA4316622

Inhibition of human BTK assessed as remaining kinase activity at 1 uM using Cdc2 peptide KVEKIGEGTYGVVYK substrate and [gamma-33P]-ATP incubated for 40 mins by radiometric protein kinase assay: 1

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
440.514.224.22
439.475.215.21
431.494.784.78
417.514.574.57
447.925.065.06
447.925.065.06
425.495.015.01
467.535.695.69
481.556.086.08
453.505.605.60
439.904.444.44
439.475.215.21
417.474.394.39
445.524.874.87
439.525.405.40
459.555.265.26
453.505.605.60
461.915.275.27
489.965.745.74
439.525.405.40
403.484.184.18
467.535.695.69
481.556.086.08
489.965.745.74
461.915.275.27
425.495.015.01
425.924.244.24
467.954.924.92