Assay Report Card

Basic Information

ID: ALA4323791

Type: Binding

Description: Negative allosteric modulation of human luteinizing hormone receptor assessed as Emax for glycoprotein human luteinizing hormone-induced agonist activity at 0.84 nM to 17 uM preincubated for 20 mins followed by 100 times EC80 of agonist addition and measured after 60 mins by cell based TR-FRET assay relative to control

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
473.946.856.85