Assay Report Card

Basic Information

ID: ALA4324375

Type: Binding

Description: Inhibition of human N- terminal His6 tagged human INMT expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL assessed as enzyme activity at 3.7 uM using tryptamine as substrate preincubated for 10 mins in presence of AdoMet followed by substrate addition by fluorescence based SAHH enzyme coupled assay relative to control

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
524.54-1.72-1.72