Assay Report Card

Basic Information

ID: ALA4324377

Type: Binding

Description: Inhibition of recombinant human His-tagged SETD7 (1 to 366 residues) expressed in Escherichia coli assessed as enzyme activity at 3.7 uM using H3-21 peptide as susbtrate preincubated for 10 mins in presence of AdoMet followed by substrate addition by fluorescence based SAHH enzyme coupled assay relative to control

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
524.54-1.72-1.72