Assay Report Card

Basic Information

ID: ALA4324384

Type: Binding

Description: Inhibition of recombinant human G9a (913 to 1193 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL assessed as enzyme activity at 11 uM using H3-21 peptide preincubated for 10 mins in presence of AdoMet followed by substrate addition by fluorescence based SAHH enzyme coupled assay relative to control

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
524.54-1.72-1.72