Agonist activity at human APJ-R expressed in HEK293 cells assessed as inhibition of forskolin- stimulated cAMP accumulation incubated for 30 mins by H...

Basic Information

ID: ALA4324418

Type: Functional

Description: Agonist activity at human APJ-R expressed in HEK293 cells assessed as inhibition of forskolin- stimulated cAMP accumulation incubated for 30 mins by HTRF assay relative to control parental HEK293 cells

Format: BAO_0000219

Organism: Homo sapiens

Cell type: HEK293

Target:  Apelin receptor(ALA1628481)

Document:  ALA4321849

Agonist activity at human APJ-R expressed in HEK293 cells assessed as inhibition of forskolin- stimulated cAMP accumulation incubated for 30 mins by HTRF assay relative to control parental HEK293 cells: 1

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
1533.83
524.027.527.52
524.027.527.52
538.057.837.83
558.996.856.85
577.016.226.22
577.016.226.22
503.607.177.17
503.607.177.17
538.057.837.83
525.016.916.91
554.057.537.53
507.577.017.01
554.057.537.53
525.007.787.78
524.027.527.52
562.985.575.57
524.027.527.52
558.478.178.17
489.586.876.87
550.068.038.03
519.606.876.87
575.047.387.38