Assay Report Card

Basic Information

ID: ALA4324995

Type: Binding

Description: Protac activity against VHL/AR in AR-positive human VCaP cells assessed as induction of AR degradation by measuring reduction in AR protein level at 100 nM incubated for 3 hrs by Western blot analysis relative to control

Organism: Homo sapiens

Cell type: VCaP

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
915.537.367.36
1095.81