Basic Information
ID: ALA4327233
Type: ADME
Description: Displacement of [3H]CP55940 from recombinant human CB1R expressed in HEK293 cell membranes at 10 uM measured after 90 mins relative to control
Format: BAO_0000219
Organism: Homo sapiens
Cell type: HEK293
Target: Cannabinoid CB1 receptor(ALA218)
Document: ALA4325860
Displacement of [3H]CP55940 from recombinant human CB1R expressed in HEK293 cell membranes at 10 uM measured after 90 mins relative to control: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA4327233
Inhibition
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 504.37 | 4.13 | 4.13 |
| 476.06 | 6.81 | 6.81 |
| 361.51 | 4.56 | 4.56 |
| 337.83 | 4.31 | 4.31 |
| 317.39 | 2.36 | 2.36 |
| 388.53 | 4.50 | 4.50 |
| 391.56 | 4.48 | 4.48 |
| 347.48 | 4.31 | 4.31 |
| 375.53 | 4.95 | 4.95 |
| 423.56 | 3.16 | 3.16 |
| 331.39 | 4.02 | 4.02 |
| 395.52 | 5.36 | 5.36 |
| 389.56 | 5.34 | 5.34 |
| 321.37 | 3.80 | 3.80 |
| 324.40 | 2.28 | 2.28 |
| 373.52 | 4.57 | 4.57 |
| 318.37 | 2.92 | 2.92 |
| 333.45 | 4.00 | 4.00 |
| 361.51 | 4.56 | 4.56 |
| 317.39 | 2.36 | 2.36 |
| 465.66 | 7.09 | 7.09 |
| 319.43 | 3.69 | 3.69 |
| 361.51 | 4.64 | 4.64 |
| 395.52 | 5.36 | 5.36 |
| 314.39 | 3.02 | 3.02 |
| 322.43 | 3.43 | 3.43 |
| 302.37 | 2.96 | 2.96 |