Basic Information
ID: ALA4329664
Type: Binding
Description: Inhibition of recombinant human C-terminal GST-tagged IKKbeta (1 to 737 residues) expressed in baculovirus expression system using GST-IkBalpha substrate measured after 30 mins by TR-FRET assay
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA4329664
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 306.37 | 3.46 | 3.46 |
| 494.66 | 3.93 | 3.93 |
| 394.50 | 3.76 | 3.76 |
| 332.40 | 4.16 | 4.16 |
| 319.36 | 2.88 | 2.88 |
| 426.54 | 2.40 | 2.40 |
| 508.69 | 4.32 | 4.32 |
| 510.66 | 3.17 | 3.17 |
| 318.38 | 3.77 | 3.77 |
| 496.63 | 2.78 | 2.78 |
| 508.69 | 4.37 | 4.37 |
| 522.72 | 4.71 | 4.71 |
| 394.50 | 3.76 | 3.76 |
| 454.60 | 3.00 | 3.00 |
| 496.68 | 4.17 | 4.17 |
| 332.40 | 4.16 | 4.16 |
| 342.42 | 2.52 | 2.52 |
| 347.42 | 3.52 | 3.52 |
| 349.43 | 3.31 | 3.31 |
| 333.39 | 3.23 | 3.23 |
| 386.45 | 3.37 | 3.37 |
| 414.50 | 4.14 | 4.14 |
| 354.43 | 2.84 | 2.84 |
| 396.51 | 4.00 | 4.00 |
| 368.46 | 3.23 | 3.23 |
| 368.46 | 3.23 | 3.23 |