Basic Information
ID: ALA4329853
Type: Binding
Description: Inhibition of recombinant human HIF-PHD1 expressed in baculovirus-infected Sf9 cells using biotin labelled DLDLEMLAPYIPMDDDFQL and 2-oxoglutarate as substrates preincubated for 30 mins followed by substrates addition and measured after 2 hrs by TR-FRET assay
Organism: Homo sapiens
Cell type: Sf9
Activity Charts
Bioactivity
Activity Types for Assay ALA4329853
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 415.43 | 1.10 | 1.10 |
| 387.37 | 0.96 | 0.96 |
| 489.36 | 2.43 | 2.43 |
| 419.34 | 0.92 | 0.92 |
| 448.36 | 2.10 | 2.10 |
| 464.42 | 3.39 | 3.39 |
| 413.31 | 0.86 | 0.86 |
| 427.34 | 0.90 | 0.90 |
| 398.29 | 0.86 | 0.86 |
| 378.77 | 1.10 | 1.10 |
| 426.35 | 1.51 | 1.51 |
| 392.80 | 1.14 | 1.14 |
| 410.38 | 1.51 | 1.51 |
| 385.33 | 0.59 | 0.59 |
| 410.39 | 0.63 | 0.63 |
| 402.40 | 0.67 | 0.67 |
| 414.30 | 0.26 | 0.26 |
| 380.30 | 0.73 | 0.73 |
| 449.34 | 1.92 | 1.92 |
| 428.32 | 1.35 | 1.35 |
| 454.79 | 3.24 | 3.24 |
| 414.30 | 0.26 | 0.26 |
| 401.35 | 0.50 | 0.50 |
| 412.32 | 1.47 | 1.47 |
| 414.30 | 0.26 | 0.26 |
| 426.35 | 1.51 | 1.51 |
| 419.34 | 0.92 | 0.92 |