Inhibition of human FLT3 at 1 uM using EAIYAAPFAKKK as substrate preincubated for 20 mins followed by [gamma-33P]-ATP addition and measured after 120 ...

Basic Information

ID: ALA4331115

Type: Binding

Description: Inhibition of human FLT3 at 1 uM using EAIYAAPFAKKK as substrate preincubated for 20 mins followed by [gamma-33P]-ATP addition and measured after 120 mins by Hotspot assay relative to control

Format: BAO_0000357

Organism: Homo sapiens

Target:  Tyrosine-protein kinase receptor FLT3(ALA1974)

Document:  ALA4330071

Inhibition of human FLT3 at 1 uM using EAIYAAPFAKKK as substrate preincubated for 20 mins followed by [gamma-33P]-ATP addition and measured after 120 mins by Hotspot assay relative to control: 1

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
391.523.493.49
449.562.812.81
420.523.183.18
455.324.314.31
369.382.272.27
432.532.422.42