Basic Information
ID: ALA4333724
Type: Binding
Description: Inhibition of kinase tracer 236 binding to recombinant full length His-tagged human CDK8/CycC expressed in baculovirus expression system preincubated for 20 mins followed by tracer addition and measured after 2 hrs by FRET-based LanthaScreen Eu kinase binding assay
Format: BAO_0000019
Organism: Homo sapiens
Target: CDK8/Cyclin C(ALA3038474)
Document: ALA4330136
Inhibition of kinase tracer 236 binding to recombinant full length His-tagged human CDK8/CycC expressed in baculovirus expression system preincubated for 20 mins followed by tracer addition and measured after 2 hrs by FRET-based LanthaScreen Eu kinase binding assay: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA4333724
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 347.44 | 4.98 | 4.98 |
| 364.42 | 4.60 | 4.60 |