Basic Information
ID: ALA4334827
Type: Binding
Description: Reversible inhibition of human immunoproteasome beta 5i subunit assessed as recovery of enzyme activity at 45 nM using Suc-LLVY-AMC as substrate preincubated for 30 mins followed by 100-fold diluted substrate addition by rapid dilution assay relative to control
Format: BAO_0000357
Organism: Homo sapiens
Target: Proteasome subunit beta type-8(ALA5620)
Document: ALA4334435
Reversible inhibition of human immunoproteasome beta 5i subunit assessed as recovery of enzyme activity at 45 nM using Suc-LLVY-AMC as substrate preincubated for 30 mins followed by 100-fold diluted substrate addition by rapid dilution assay relative to control: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA4334827
Activity
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 640.76 | 4.68 | 4.68 |