Inhibition of human immunoproteasome beta 5i subunit using Suc-LLVY-AMC as substrate assessed as residual activity at 10 uM preincubated for 30 mins f...

Basic Information

ID: ALA4334843

Type: Binding

Description: Inhibition of human immunoproteasome beta 5i subunit using Suc-LLVY-AMC as substrate assessed as residual activity at 10 uM preincubated for 30 mins followed by substrate addition measured for 120 mins by fluorescence based assay relative to control

Format: BAO_0000357

Organism: Homo sapiens

Target:  Proteasome subunit beta type-8(ALA5620)

Document:  ALA4334435

Inhibition of human immunoproteasome beta 5i subunit using Suc-LLVY-AMC as substrate assessed as residual activity at 10 uM preincubated for 30 mins followed by substrate addition measured for 120 mins by fluorescence based assay relative to control: 1

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
392.464.424.42
378.434.084.08
437.454.054.05
406.484.814.81
392.464.474.47