Assay Report Card

Basic Information

ID: ALA4334957

Type: Binding

Description: Inhibition of human ABL1 Y253F mutant (27 to end residues) assessed as residual activity at 1 uM using EAIYAAPFAKKK as substrate incubated for 40 mins in presence of [gamma-33ATP] by scintillation counting based radiometry assay relative to control

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
315.312.992.99
388.833.293.29