Basic Information
ID: ALA4337392
Type: Binding
Description: Displacement of 20 nM [3H]UR-DE257 from human H2R expressed in Sf9 cell membranes co-expressing GsalphaS by competition binding assay
Organism: Homo sapiens
Cell type: Sf9
Activity Charts
Bioactivity
Activity Types for Assay ALA4337392
Ki
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 465.40 | 1.70 | 1.70 |
| 505.46 | 2.07 | 2.07 |
| 491.43 | 1.73 | 1.73 |
| 519.45 | 1.00 | 1.00 |
| 514.43 | 2.22 | 2.22 |
| 477.41 | 1.47 | 1.47 |
| 562.54 | 3.31 | 3.31 |
| 516.44 | 2.70 | 2.70 |
| 533.47 | 1.34 | 1.34 |
| 502.42 | 2.31 | 2.31 |
| 491.43 | 2.10 | 2.10 |
| 477.41 | 1.34 | 1.34 |
| 491.43 | 1.73 | 1.73 |
| 491.43 | 1.69 | 1.69 |
| 419.45 | 2.04 | 2.04 |
| 505.46 | 2.08 | 2.08 |
| 477.41 | 1.71 | 1.71 |
| 634.50 | 1.02 | 1.02 |
| 519.45 | 0.95 | 0.95 |
| 451.37 | 1.31 | 1.31 |