Basic Information
ID: ALA4337395
Type: Binding
Description: Selectivity index, ratio of Ki for displacement of 2 nM [3H]UR-PI294 from human H3R expressed in Sf9 cell membranes co-expressing Gia2 and beta1gamma2 by competition binding assay to Ki for displacement of 40 nM [3H]-histamine from human H4R expressed in Sf9 cell membranes co-expressing Gia2 and beta1gamma2 by competition binding assay
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA4337395
Ratio Ki
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 465.40 | 1.70 | 1.70 |
| 491.43 | 1.73 | 1.73 |
| 519.45 | 1.00 | 1.00 |
| 516.44 | 2.70 | 2.70 |
| 502.42 | 2.31 | 2.31 |
| 491.43 | 2.10 | 2.10 |
| 491.43 | 1.73 | 1.73 |
| 419.45 | 2.04 | 2.04 |
| 477.41 | 1.71 | 1.71 |