Assay Report Card

Basic Information

ID: ALA4337397

Type: Binding

Description: Selectivity index, ratio of Ki for [3H]UR-DE257 from human H2R expressed in Sf9 cell membranes co-expressing GsalphaS by competition binding assay to Ki for displacement of 40 nM [3H]-histamine from human H4R expressed in Sf9 cell membranes co-expressing Gia2 and beta1gamma2 by competition binding assay

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
465.401.701.70
491.431.731.73
519.451.001.00
491.432.102.10
491.431.731.73
419.452.042.04
477.411.711.71