ID: ALA4338950
Type: Binding
Description: Inhibition of recombinant N-terminal FLAG/His-tagged SMYD3 (unknown origin) expressed in baculovirus infected insect cells using 3H-SAM as substrate assessed as 3H-MEKK2 methylation incubated for 40 mins by scintillation proximity assay
Organism: Homo sapiens
Bioactivity
Activity Types for Assay ALA4338950
IC50
Parent Molecular Weight | ALogP | Polar Surface Area |
---|---|---|
432.55 | 2.20 | 2.20 |
396.51 | 1.35 | 1.35 |
480.68 | 3.27 | 3.27 |
472.61 | 3.12 | 3.12 |
501.65 | 2.82 | 2.82 |
534.65 | 3.91 | 3.91 |
501.65 | 2.82 | 2.82 |
327.41 | 1.10 | 1.10 |
519.64 | 2.96 | 2.96 |
438.59 | 2.20 | 2.20 |
520.62 | 3.57 | 3.57 |
313.38 | 0.71 | 0.71 |
535.11 | 4.08 | 4.08 |
500.67 | 3.42 | 3.42 |
342.42 | 0.03 | 0.03 |
519.64 | 2.96 | 2.96 |
518.66 | 3.56 | 3.56 |
452.62 | 2.63 | 2.63 |
506.59 | 3.32 | 3.32 |
444.56 | 2.34 | 2.34 |
518.66 | 3.56 | 3.56 |
410.54 | 1.59 | 1.59 |
501.65 | 2.82 | 2.82 |
514.69 | 3.73 | 3.73 |
514.69 | 3.73 | 3.73 |
382.49 | 0.83 | 0.83 |
458.58 | 2.73 | 2.73 |
410.54 | 1.56 | 1.56 |
438.59 | 2.24 | 2.24 |
370.48 | 0.81 | 0.81 |
536.10 | 3.47 | 3.47 |
519.64 | 2.96 | 2.96 |
368.46 | 0.44 | 0.44 |
396.51 | 1.17 | 1.17 |
535.11 | 4.08 | 4.08 |
548.67 | 4.30 | 4.30 |
466.65 | 2.88 | 2.88 |
466.65 | 3.02 | 3.02 |
396.51 | 1.35 | 1.35 |
535.11 | 4.08 | 4.08 |
404.49 | 1.59 | 1.59 |
514.69 | 3.73 | 3.73 |
494.70 | 3.66 | 3.66 |
506.59 | 3.18 | 3.18 |
410.54 | 1.59 | 1.59 |
515.68 | 3.13 | 3.13 |
424.57 | 1.85 | 1.85 |
410.54 | 1.56 | 1.56 |
518.66 | 3.56 | 3.56 |