Assay Report Card

Basic Information

ID: ALA4339642

Type: Binding

Description: Negative allosteric modulation of rat GABAA alpha1beta2gamma2S expressed in Xenopus laevis oocytes assessed as inhibition of GABA-induced current response at 30 uM at -40 mV holding potential by two-electrode voltage clamp method relative to GABA alone

Organism: Rattus norvegicus

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
495.604.304.30
351.414.264.26