Assay Report Card

Basic Information

ID: ALA4339646

Type: Binding

Description: Negative allosteric modulation of rat alpha1betagammadelta nACHR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response at 30 uM at -40 mV holding potential by two-electrode voltage clamp method relative to acetylcholine alone

Organism: Rattus norvegicus

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
495.604.304.30
351.414.264.26