Assay Report Card

Basic Information

ID: ALA4339875

Type: Binding

Description: Inhibition of rat DYRK1A kinase domain (1 to 499 residues) expressed in bacteria assessed as residual activity at 1 uM using KKISGRLSPIMTEQ as substrate in presence of [gamma33P]ATP relative to control

Organism: Rattus norvegicus

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
241.211.671.67
352.403.863.86
296.292.312.31
298.312.022.02
354.413.573.57