Basic Information
ID: ALA4339875
Type: Binding
Description: Inhibition of rat DYRK1A kinase domain (1 to 499 residues) expressed in bacteria assessed as residual activity at 1 uM using KKISGRLSPIMTEQ as substrate in presence of [gamma33P]ATP relative to control
Format: BAO_0000019
Organism: Rattus norvegicus
Target: Dual specificity tyrosine-phosphorylation-regulated kinase 1A(ALA5508)
Document: ALA4339207
Inhibition of rat DYRK1A kinase domain (1 to 499 residues) expressed in bacteria assessed as residual activity at 1 uM using KKISGRLSPIMTEQ as substrate in presence of [gamma33P]ATP relative to control: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA4339875
Activity
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 241.21 | 1.67 | 1.67 |
| 352.40 | 3.86 | 3.86 |
| 296.29 | 2.31 | 2.31 |
| 298.31 | 2.02 | 2.02 |
| 354.41 | 3.57 | 3.57 |