Basic Information
ID: ALA4341001
Type: Binding
Description: Selectivity index, ratio of IC50 for inhibition of human ERG incubated for 1 hr by fluorescence polarization binding assay to IC50 for inhibition of His tagged human recombinant PIM1 using PIM tide (ARKRRRHPSGPPTA) as substrate incubated for 1 hr by fluorescence based assay
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA4341001
Ratio IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 422.41 | 3.13 | 3.13 |
| 405.42 | 4.05 | 4.05 |
| 414.51 | 4.52 | 4.52 |
| 448.51 | 2.67 | 2.67 |
| 430.52 | 2.67 | 2.67 |
| 482.95 | 3.33 | 3.33 |
| 415.50 | 3.91 | 3.91 |
| 484.49 | 2.95 | 2.95 |
| 466.50 | 2.81 | 2.81 |
| 444.54 | 2.92 | 2.92 |
| 415.50 | 3.91 | 3.91 |
| 474.57 | 2.60 | 2.60 |
| 448.51 | 2.67 | 2.67 |