Assay Report Card

Basic Information

ID: ALA4341032

Type: Binding

Description: Bias factor, change in deltalog(Tau/KA) for agonist activity at Rluc-tagged MOR receptor (unknown origin) expressed in human SH-5YSY cells co-expressing RGFP-fused to Gbeta1 assessed as increase in MOR/G beta1 protein interaction incubated for 5 mins in presence of coelenterazine by BRET assay to deltalog(Tau/KA) for agonist activity at Rluc-tagged MOR receptor (unknown origin) expressed in human SH-5YSY cells co-expressing RGFP-fused to MOR/beta-arrestin-2 assessed as increase in beta-arrestin-2 protein interaction incubated for 5 mins in presence of coelenterazine by BRET assay

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
569.660.230.23
351.494.304.30
351.494.304.30