Basic Information
ID: ALA4341809
Type: Binding
Description: Inhibition of wild type HIV1 protease expressed in Escherichia coli using Arg-Glu (EDANS)-Ser-Gln-Asn-Tyr-Pro-Ile-Val-Gln-Lys(DABCYL)-Arg as substrate preincubated for 20 to 30 mins followed by substrate addition and measured for 10 mins by FRET assay
Organism: Human immunodeficiency virus 1
Activity Charts
Bioactivity
Activity Types for Assay ALA4341809
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 547.67 | 2.38 | 2.38 |
| 596.67 | 1.75 | 1.75 |
| 596.67 | 1.75 | 1.75 |
| 601.13 | 2.08 | 2.08 |
| 551.67 | 1.84 | 1.84 |
| 565.70 | 2.15 | 2.15 |
| 611.68 | 2.18 | 2.18 |
| 581.70 | 1.85 | 1.85 |
| 586.12 | 2.50 | 2.50 |
| 567.67 | 1.55 | 1.55 |
| 631.12 | 2.41 | 2.41 |
| 626.70 | 1.76 | 1.76 |
| 565.70 | 2.15 | 2.15 |
| 566.69 | 1.43 | 1.43 |
| 597.65 | 1.88 | 1.88 |
| 595.68 | 2.48 | 2.48 |
| 612.67 | 1.46 | 1.46 |
| 580.71 | 2.58 | 2.58 |
| 566.68 | 2.27 | 2.27 |
| 596.71 | 2.28 | 2.28 |
| 616.10 | 2.82 | 2.82 |
| 581.70 | 1.85 | 1.85 |
| 611.73 | 1.86 | 1.86 |
| 597.70 | 1.56 | 1.56 |
| 582.69 | 1.13 | 1.13 |
| 580.71 | 2.58 | 2.58 |
| 595.68 | 2.48 | 2.48 |
| 582.68 | 1.98 | 1.98 |
| 581.66 | 2.17 | 2.17 |
| 581.70 | 1.85 | 1.85 |
| 596.71 | 1.43 | 1.43 |
| 601.13 | 2.92 | 2.92 |
| 566.69 | 1.43 | 1.43 |
| 616.14 | 2.51 | 2.51 |