Assay Report Card

Basic Information

ID: ALA4342201

Type: Binding

Description: Inhibition of NO711 binding to mouse GAT1 expressed in HEK293 cell membranes assessed as residual binding at 1 uM incubated for 4 hrs in presence of NO711 by LC-ESI-MS/MS analysis relative to control

Organism: Mus musculus

Cell type: HEK293

Activity Charts

Bioactivity

Activity Types for Assay ALA4342201

Activity

Total(247)

Compound Summary

Parent Molecular Weight	ALogP	Polar Surface Area
107.11	0.89	0.89
107.11	0.89	0.89
122.12	1.20	1.20
152.15	1.21	1.21
106.12	1.50	1.50
136.15	1.51	1.51
198.22	3.29	3.29
132.16	1.90	1.90
212.25	3.08	3.08
212.25	3.08	3.08
112.15	1.56	1.56
122.12	1.20	1.20
182.22	3.17	3.17
182.22	3.17	3.17
182.22	3.17	3.17
251.11	4.47	4.47
136.15	1.51	1.51
151.12	1.41	1.41
151.12	1.41	1.41
96.08	1.09	1.09
120.15	1.81	1.81
206.63	3.41	3.41
182.17	1.22	1.22
136.15	1.51	1.51
162.23	2.80	2.80
140.57	2.15	2.15
151.12	1.41	1.41
150.13	1.23	1.23
162.21	2.71	2.71
251.62	3.32	3.32
120.15	1.43	1.43
157.17	2.05	2.05
146.15	1.38	1.38
198.22	3.29	3.29
175.01	2.81	2.81
120.15	1.81	1.81
204.31	3.36	3.36
140.57	2.15	2.15
256.18	3.66	3.66
157.17	2.05	2.05
172.19	1.68	1.68
131.13	1.37	1.37
198.22	3.29	3.29
95.10	0.83	0.83
107.11	0.89	0.89
156.18	2.65	2.65
200.21	3.31	3.31
200.21	3.31	3.31
200.21	3.31	3.31
218.20	3.44	3.44
218.20	3.44	3.44
218.20	3.44	3.44
218.20	3.44	3.44
218.20	3.44	3.44
230.24	3.31	3.31
230.24	3.31	3.31
230.24	3.31	3.31
212.25	3.17	3.17
216.67	3.82	3.82
216.67	3.82	3.82
216.67	3.82	3.82
212.25	3.17	3.17
212.25	3.17	3.17
196.25	3.47	3.47
196.25	3.47	3.47
200.21	3.31	3.31
200.21	3.31	3.31
234.66	3.96	3.96
251.11	4.47	4.47
218.20	3.44	3.44
236.19	3.58	3.58
218.20	3.44	3.44
234.66	3.96	3.96
196.25	3.47	3.47
210.28	3.78	3.78
318.22	5.20	5.20
234.66	3.96	3.96
258.32	4.83	4.83
258.32	4.83	4.83
234.66	3.96	3.96
258.32	4.83	4.83
174.98	1.85	1.85
124.11	1.64	1.64
149.19	1.57	1.57
185.02	2.26	2.26
156.18	2.65	2.65
201.22	2.77	2.77
134.18	1.99	1.99
185.02	2.26	2.26
188.25	3.23	3.23
124.11	1.64	1.64
124.11	1.64	1.64
414.51	4.78	4.78
150.13	1.23	1.23
216.67	3.82	3.82
217.66	3.21	3.21
205.64	3.01	3.01
177.23	2.35	2.35
244.22	3.03	3.03
386.42	3.26	3.26
295.12	4.20	4.20
200.21	3.31	3.31
186.01	1.66	1.66
186.01	1.66	1.66
171.20	2.29	2.29
201.20	2.70	2.70
201.20	2.70	2.70
213.24	2.57	2.57
217.66	3.21	3.21
202.28	3.54	3.54
217.66	3.21	3.21
356.40	3.25	3.25
240.18	3.78	3.78
206.24	3.81	3.81
224.23	3.51	3.51
206.24	3.81	3.81
188.25	3.23	3.23
186.21	2.66	2.66
206.24	3.37	3.37
202.28	3.54	3.54
269.10	4.61	4.61
174.17	2.79	2.79
230.29	2.58	2.58
188.25	3.23	3.23
232.28	4.32	4.32
186.21	1.90	1.90
184.20	1.96	1.96
217.66	3.21	3.21
356.40	3.25	3.25
170.21	2.96	2.96
234.26	3.11	3.11
171.20	2.49	2.49
324.24	5.27	5.27
222.70	3.88	3.88
183.21	2.56	2.56
202.28	3.54	3.54
197.24	2.87	2.87
258.17	3.92	3.92
386.42	3.26	3.26
407.30	4.42	4.42
154.60	2.08	2.08
202.28	3.54	3.54
190.23	2.02	2.02
206.63	3.41	3.41
172.18	2.36	2.36
216.67	3.82	3.82
191.23	1.28	1.28
199.21	1.54	1.54
239.20	3.31	3.31
274.62	4.43	4.43
251.08	3.52	3.52
352.43	3.42	3.42
251.08	3.52	3.52
219.67	3.16	3.16
390.84	3.90	3.90
209.23	1.37	1.37
184.20	1.96	1.96
338.41	3.11	3.11
196.25	3.02	3.02
240.26	2.94	2.94
392.38	3.53	3.53
150.18	1.40	1.40
234.26	3.11	3.11
162.15	1.48	1.48
190.12	2.40	2.40
186.01	1.66	1.66
308.18	4.80	4.80
244.25	1.97	1.97
222.70	3.88	3.88
192.11	2.66	2.66
108.10	0.29	0.29
226.23	2.89	2.89
374.39	3.39	3.39
374.39	3.39	3.39
222.70	3.88	3.88
188.25	3.23	3.23
374.39	3.39	3.39
131.13	1.37	1.37
201.20	2.70	2.70
188.19	1.86	1.86
252.10	3.87	3.87
390.84	3.90	3.90
257.14	4.53	4.53
272.35	4.22	4.22
206.63	3.41	3.41
183.21	2.56	2.56
212.27	2.96	2.96
221.64	3.12	3.12
221.98	1.70	1.70
186.01	1.66	1.66
174.12	2.52	2.52
183.21	2.56	2.56
194.23	3.07	3.07
202.19	2.10	2.10
190.18	2.03	2.03
120.15	1.81	1.81
390.84	3.90	3.90
374.39	3.39	3.39
213.24	1.90	1.90
250.22	4.18	4.18
201.20	2.70	2.70
217.66	3.21	3.21
216.31	3.84	3.84
172.18	2.76	2.76
202.28	3.54	3.54
224.62	3.55	3.55
174.16	1.55	1.55
222.33	3.91	3.91
366.46	3.73	3.73
172.18	2.76	2.76
174.98	1.85	1.85
190.12	2.40	2.40
241.07	4.07	4.07
326.32	4.64	4.64
190.12	2.40	2.40
362.43	4.25	4.25
192.11	2.66	2.66
374.39	3.39	3.39
154.60	2.08	2.08
122.17	1.40	1.40
174.12	2.52	2.52
216.67	3.82	3.82
390.84	3.90	3.90
251.11	4.47	4.47
240.18	3.78	3.78
232.28	4.32	4.32
154.60	2.08	2.08
222.24	3.91	3.91
186.01	1.66	1.66
196.25	3.09	3.09
174.12	2.52	2.52
131.13	1.37	1.37
274.62	4.43	4.43
414.51	4.78	4.78
414.51	4.78	4.78
260.68	3.55	3.55
140.57	2.15	2.15
386.42	3.26	3.26
212.25	2.12	2.12
229.03	1.99	1.99
175.01	2.81	2.81
202.28	3.54	3.54
214.22	1.96	1.96
474.40	5.15	5.15
185.19	1.35	1.35
222.70	3.88	3.88
374.39	3.39	3.39