Basic Information
ID: ALA4344212
Type: Binding
Description: Antagonist activity at human Gi/o-coupled CNR1 expressed in CHOK1 cells assessed as inhibition in CP55940-induced beta-arrestin 2 recruitment incubated for 30 mins followed by CP55940 addition and measured after 90 or 180 mins by pathhunter beta-arrestin assay
Format: BAO_0000219
Organism: Homo sapiens
Target: Cannabinoid CB1 receptor(ALA218)
Document: ALA4342456
Antagonist activity at human Gi/o-coupled CNR1 expressed in CHOK1 cells assessed as inhibition in CP55940-induced beta-arrestin 2 recruitment incubated for 30 mins followed by CP55940 addition and measured after 90 or 180 mins by pathhunter beta-arrestin assay: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA4344212
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 509.44 | 6.01 | 6.01 |