Basic Information
ID: ALA4344230
Type: Binding
Description: Antagonist activity at human Gq-coupled PRLHR expressed in CHOK1 cells assessed as inhibition in prolactin releasing peptide (1 to 31)-induced beta-arrestin 2 recruitment incubated for 30 mins followed by prolactin releasing peptide (1 to 31) addition and measured after 90 or 180 mins by pathhunter beta-arrestin assay
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA4344230
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 509.44 | 6.01 | 6.01 |
| 561.48 | 5.42 | 5.42 |