Basic Information
ID: ALA4344232
Type: Binding
Description: Antagonist activity at human Gq-coupled HCRTR2 expressed in CHOK1 cells assessed as inhibition in Orexin A-induced beta-arrestin 2 recruitment incubated for 30 mins followed by Orexin A addition and measured after 90 or 180 mins by pathhunter beta-arrestin assay
Format: BAO_0000219
Organism: Homo sapiens
Target: Orexin receptor 2(ALA4792)
Document: ALA4342456
Antagonist activity at human Gq-coupled HCRTR2 expressed in CHOK1 cells assessed as inhibition in Orexin A-induced beta-arrestin 2 recruitment incubated for 30 mins followed by Orexin A addition and measured after 90 or 180 mins by pathhunter beta-arrestin assay: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA4344232
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 480.62 | 4.44 | 4.44 |