Basic Information
ID: ALA4345336
Type: Binding
Description: Antagonist activity at C-terminal RLuc8-fused D1R (unknown origin) transfected in human HEK293T cells co-expressing N-terminal Venus-tagged beta-arrestin2 assessed as increase in beta-arrestin2 recruitment measured after 5 mins in presence of coelenterazine H by BRET assay
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA4345336
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 287.79 | 3.67 | 3.67 |
| 323.44 | 4.02 | 4.02 |
| 323.44 | 4.02 | 4.02 |
| 374.28 | 4.22 | 4.22 |
| 374.28 | 4.22 | 4.22 |
| 374.28 | 4.22 | 4.22 |
| 374.28 | 4.22 | 4.22 |
| 309.41 | 3.76 | 3.76 |