Basic Information
ID: ALA4346471
Type: Binding
Description: Activation of recombinant EPAC1 (149 to 881 residues) (unknown origin) assessed as stimulation of dissociation of fluorescent MANT-GDP from recombinant Rap1b in presence of excess nonfluorescent nucleotides by fluorescence based in-vitro GEF assay
Format: BAO_0000357
Organism: Homo sapiens
Target: Rap guanine nucleotide exchange factor 3(ALA2029197)
Document: ALA4342525
Activation of recombinant EPAC1 (149 to 881 residues) (unknown origin) assessed as stimulation of dissociation of fluorescent MANT-GDP from recombinant Rap1b in presence of excess nonfluorescent nucleotides by fluorescence based in-vitro GEF assay: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA4346471
EC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 401.44 | 2.74 | 2.74 |
| 416.46 | 2.32 | 2.32 |
| 421.47 | 3.89 | 3.89 |