Basic Information
ID: ALA4346474
Type: Binding
Description: Activation of recombinant EPAC1 (149 to 881 residues) (unknown origin) assessed as stimulation of dissociation of fluorescent MANT-GDP from recombinant Rap1b at 10 uM in presence of excess nonfluorescent nucleotides by fluorescence based in-vitro GEF assay relative to cAMP
Format: BAO_0000357
Organism: Homo sapiens
Target: Rap guanine nucleotide exchange factor 3(ALA2029197)
Document: ALA4342525
Activation of recombinant EPAC1 (149 to 881 residues) (unknown origin) assessed as stimulation of dissociation of fluorescent MANT-GDP from recombinant Rap1b at 10 uM in presence of excess nonfluorescent nucleotides by fluorescence based in-vitro GEF assay relative to cAMP: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA4346474
Activity
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 401.44 | 2.74 | 2.74 |
| 515.51 | 5.19 | 5.19 |
| 374.39 | 2.44 | 2.44 |
| 416.46 | 2.32 | 2.32 |
| 404.38 | 2.77 | 2.77 |
| 421.47 | 3.89 | 3.89 |