Assay Report Card

Basic Information

ID: ALA4346474

Type: Binding

Description: Activation of recombinant EPAC1 (149 to 881 residues) (unknown origin) assessed as stimulation of dissociation of fluorescent MANT-GDP from recombinant Rap1b at 10 uM in presence of excess nonfluorescent nucleotides by fluorescence based in-vitro GEF assay relative to cAMP

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
401.442.742.74
515.515.195.19
374.392.442.44
416.462.322.32
404.382.772.77
421.473.893.89