Assay Report Card

Basic Information

ID: ALA4350283

Type: Binding

Description: Inhibition of N-terminal GST tagged human recombinant EHMT1 (794 to 1294 residues) expressed in baculovirus infected Sf9 insect cells assessed as reduction in conversion of SAH to AMP using histone H3 as substrate and SAH as cosubstrate incubated for 30 mins by AMP Glo detection assay

Organism: Homo sapiens

Cell type: Sf9

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
485.682.622.62
509.745.845.84
329.442.982.98
463.674.884.88
498.681.581.58
495.723.493.49
461.613.353.35
427.614.994.99
439.654.864.86
499.661.761.76
441.622.182.18
495.723.363.36
426.613.243.24
384.532.292.29
467.663.103.10
498.681.761.76
496.661.331.33
479.631.771.77
480.704.724.72
509.702.842.84
469.682.782.78
499.702.142.14
495.723.313.31
552.772.892.89
489.673.473.47
437.591.601.60
461.613.353.35
451.621.991.99
495.671.561.56
470.621.571.57
507.725.535.53
477.705.275.27
427.551.391.39
435.624.284.28
485.643.083.08
461.613.353.35
483.662.362.36
470.620.970.97
505.672.262.26
472.126.116.11
495.723.223.22
509.745.245.24
468.694.944.94
455.675.605.60
503.694.944.94
423.584.414.41
412.582.852.85
498.682.352.35
467.705.475.47
468.674.854.85
467.662.752.75
465.695.445.44
465.652.202.20
451.621.861.86
484.651.371.37
460.633.953.95
481.735.865.86
498.682.182.18
491.682.732.73